Full Kinase Panel
Through our partner Carna Biosciences we are offering the Full Kinase Panel. This panel is comprised of all the kinase assays available at Carna Biosciences, currently more than 300 assays. Clients can either choose to run the full panel or can ‘cherry-pick’ their most preferred kinases.
Kinases Available in the Full Kinase panel
The Full Kinase Panel -available at Carna- enables clients to extensively profile their compounds on almost the entire kinome. The full kinase panel is run with high accuracy and a rapid turn-around time of 4 weeks with intermediate reporting at 2 weeks.
Target Name |
Group |
Assay Type |
Source (Carna Cat No.) |
ABL (ABL1) |
TK |
Mobility Shift, IMAPTM |
08-001 |
ABL (ABL1) [E255K] |
TK |
Mobility Shift, IMAPTM |
08-094 |
ABL (ABL1) [T315I] |
TK |
Mobility Shift, IMAPTM |
08-093 |
ACK (TNK2) |
TK |
Mobility Shift, IMAPTM |
08-196 |
AKT1 |
STK |
Mobility Shift, IMAPTM |
01-101 |
AKT2 |
STK |
Mobility Shift, IMAPTM |
01-102 |
AKT3 |
STK |
Mobility Shift, IMAPTM |
01-103 |
ALK |
TK |
Mobility Shift, IMAPTM |
08-518 |
ALK[F1174L] |
TK |
Mobility Shift, IMAPTM |
08-519 |
ALK[L1196M] |
TK |
Mobility Shift, IMAPTM |
08-529 |
ALK[R1275Q] |
TK |
Mobility Shift, IMAPTM |
08-520 |
AMPKα1/β1/γ1 (PRKAA1/B1/G1) |
STK |
Mobility Shift, IMAPTM |
02-113 |
AMPKα2/β1/γ1 (PRKAA2/B1/G1) |
STK |
Mobility Shift, IMAPTM |
02-114 |
ARG (ABL2) |
TK |
Mobility Shift, IMAPTM |
08-102 |
AurA (AURKA) |
STK |
Mobility Shift, IMAPTM |
05-101 |
AurA(AURKA)/TPX2 |
STK |
Mobility Shift, IMAPTM |
05-186 |
AurB (AURKB)/INCENP |
STK |
Mobility Shift, IMAPTM |
05-102 |
AurC (AURKC) |
STK |
Mobility Shift, IMAPTM |
05-103 |
AXL |
TK |
Mobility Shift, IMAPTM |
08-107 |
BLK |
TK |
Mobility Shift, IMAPTM |
08-164 |
BMPR1A |
STK |
ELISA |
09-137 |
BMX |
TK |
Mobility Shift, IMAPTM |
08-179 |
BRAF |
STK |
ELISA |
09-122 |
BRAF |
STK |
Mobility Shift, IMAPTM |
09-122 |
BRAF [V600E] |
STK |
ELISA |
09-144 |
BRAF[V600E] |
STK |
Mobility Shift, IMAPTM |
09-144 |
BRK (PTK6) |
TK |
Mobility Shift, IMAPTM |
08-165 |
BRSK1 |
STK |
Mobility Shift, IMAPTM |
02-115 |
BRSK2 |
STK |
Mobility Shift, IMAPTM |
02-116 |
BTK |
TK |
Mobility Shift, IMAPTM |
08-080 |
CaMK1α (CAMK1) |
STK |
Mobility Shift, IMAPTM |
02-104 |
CaMK1δ (CAMK1D) |
STK |
Mobility Shift, IMAPTM |
02-106 |
CaMK2α (CAMK2A) |
STK |
Mobility Shift, IMAPTM |
02-109 |
CaMK2β (CAMK2B) |
STK |
Mobility Shift, IMAPTM |
02-110 |
CaMK2γ (CAMK2G) |
STK |
Mobility Shift, IMAPTM |
02-112 |
CaMK2δ (CAMK2D) |
STK |
Mobility Shift, IMAPTM |
02-111 |
CaMK4 |
STK |
Mobility Shift, IMAPTM |
02-108 |
CDC2 /CycB1 |
STK |
Mobility Shift, IMAPTM |
04-102 |
CDC7/ASK |
STK |
Mobility Shift, IMAPTM |
05-109 |
CDK2 /CycA2 |
STK |
Mobility Shift, IMAPTM |
04-103 |
CDK2 /CycE1 |
STK |
Mobility Shift, IMAPTM |
04-165 |
CDK3 /CycE1 |
STK |
Mobility Shift, IMAPTM |
04-104 |
CDK4 /CycD3 |
STK |
Mobility Shift, IMAPTM |
04-105 |
CDK5 /p25 |
STK |
Mobility Shift, IMAPTM |
04-106 |
CDK6 /CycD3 |
STK |
Mobility Shift, IMAPTM |
04-107 |
CDK7 /CycH/MAT1 |
STK |
Mobility Shift, IMAPTM |
04-108 |
CDK9 /CycT1 |
STK |
Mobility Shift, IMAPTM |
04-110 |
CGK2 (PRKG2) |
STK |
Mobility Shift, IMAPTM |
01-143 |
CHK1 (CHEK1) |
STK |
Mobility Shift, IMAPTM |
02-117 |
CHK2 (CHEK2) |
STK |
Mobility Shift, IMAPTM |
02-162 |
CK1α (CSNK1A1) |
STK |
Mobility Shift, IMAPTM |
03-101 |
CK1γ1 (CSNK1G1) |
STK |
Mobility Shift, IMAPTM |
03-105 |
CK1γ2 (CSNK1G2) |
STK |
Mobility Shift, IMAPTM |
03-106 |
CK1γ3 (CSNK1G3) |
STK |
Mobility Shift, IMAPTM |
03-107 |
CK1δ (CSNK1D) |
STK |
Mobility Shift, IMAPTM |
03-103 |
CK1ε (CSNK1E) |
STK |
Mobility Shift, IMAPTM |
03-104 |
CK2α1/β (CSNK2A1/B) |
STK |
Mobility Shift, IMAPTM |
05-184 |
CK2α2/β (CSNK2A2/B) |
STK |
Mobility Shift, IMAPTM |
05-185 |
CLK1 |
STK |
Mobility Shift, IMAPTM |
04-126 |
CLK2 |
STK |
Mobility Shift, IMAPTM |
04-127 |
CLK3 |
STK |
Mobility Shift, IMAPTM |
04-128 |
COT (MAP3K8) |
STK |
Mobility Shift, IMAPTM |
07-301 |
COT(MAP3K8) |
STK |
ELISA |
07-301 |
CRIK (CIT) |
STK |
Mobility Shift, IMAPTM |
01-104 |
CSK |
TK |
Mobility Shift, IMAPTM |
08-111 |
DAPK1 |
STK |
Mobility Shift, IMAPTM |
02-134 |
DCAMKL2 |
STK |
Mobility Shift, IMAPTM |
02-140 |
DDR1 |
TK |
Mobility Shift, IMAPTM |
08-113 |
DDR2 |
TK |
Mobility Shift, IMAPTM |
08-114 |
DLK (MAP3K12) |
STK |
Mobility Shift, IMAPTM |
09-111 |
DLK(MAP3K12) |
STK |
ELISA |
09-111 |
DYRK1A |
STK |
Mobility Shift, IMAPTM |
04-130 |
DYRK1B |
STK |
Mobility Shift, IMAPTM |
04-131 |
DYRK2 |
STK |
Mobility Shift, IMAPTM |
04-132 |
DYRK3 |
STK |
Mobility Shift, IMAPTM |
04-133 |
EEF2K |
STK |
Mobility Shift, IMAPTM |
10-113 |
EGFR |
TK |
Mobility Shift, IMAPTM |
08-115 |
EGFR[d746-750/T790M] |
TK |
Mobility Shift, IMAPTM |
08-528 |
EGFR[d746-750] |
TK |
Mobility Shift, IMAPTM |
08-527 |
EGFR[L858R] |
TK |
Mobility Shift, IMAPTM |
08-502 |
EGFR[L861Q] |
TK |
Mobility Shift, IMAPTM |
08-513 |
EGFR[T790M/L858R] |
TK |
Mobility Shift, IMAPTM |
08-510 |
EGFR[T790M] |
TK |
Mobility Shift, IMAPTM |
08-194 |
EML4-ALK |
TK |
Mobility Shift, IMAPTM |
08-516 |
EPHA1 |
TK |
Mobility Shift, IMAPTM |
08-119 |
EPHA2 |
TK |
Mobility Shift, IMAPTM |
08-121 |
EPHA3 |
TK |
Mobility Shift, IMAPTM |
08-122 |
EPHA4 |
TK |
Mobility Shift, IMAPTM |
08-123 |
EPHA5 |
TK |
Mobility Shift, IMAPTM |
08-124 |
EPHA6 |
TK |
Mobility Shift, IMAPTM |
08-125 |
EPHA7 |
TK |
Mobility Shift, IMAPTM |
08-126 |
EPHA8 |
TK |
Mobility Shift, IMAPTM |
08-127 |
EPHB1 |
TK |
Mobility Shift, IMAPTM |
08-128 |
EPHB2 |
TK |
Mobility Shift, IMAPTM |
08-129 |
EPHB3 |
TK |
Mobility Shift, IMAPTM |
08-130 |
EPHB4 |
TK |
Mobility Shift, IMAPTM |
08-131 |
Erk1 (MAPK3) |
STK |
Mobility Shift, IMAPTM |
04-142 |
Erk2 (MAPK1) |
STK |
Mobility Shift, IMAPTM |
04-143 |
Erk5 (MAPK7) |
STK |
Mobility Shift, IMAPTM |
04-146 |
FAK (PTK2) |
TK |
Mobility Shift, IMAPTM |
08-137 |
FER |
TK |
Mobility Shift, IMAPTM |
08-139 |
FES |
TK |
Mobility Shift, IMAPTM |
08-140 |
FGFR1 |
TK |
Mobility Shift, IMAPTM |
08-133 |
FGFR1[V561M] |
TK |
Mobility Shift, IMAPTM |
08-536 |
FGFR2 |
TK |
Mobility Shift, IMAPTM |
08-134 |
FGFR3 |
TK |
Mobility Shift, IMAPTM |
08-135 |
FGFR3[K650E] |
TK |
Mobility Shift, IMAPTM |
08-501 |
FGFR3[K650M] |
TK |
Mobility Shift, IMAPTM |
08-199 |
FGFR4 |
TK |
Mobility Shift, IMAPTM |
08-136 |
FGFR4[N535K] |
TK |
Mobility Shift, IMAPTM |
08-524 |
FGFR4[V550E] |
TK |
Mobility Shift, IMAPTM |
08-525 |
FGFR4[V550L] |
TK |
Mobility Shift, IMAPTM |
08-526 |
FGR |
TK |
Mobility Shift, IMAPTM |
08-166 |
FLT1 |
TK |
Mobility Shift, IMAPTM |
08-189 |
FLT3 |
TK |
Mobility Shift, IMAPTM |
08-154 |
FLT4 |
TK |
Mobility Shift, IMAPTM |
08-190 |
FMS (CSF1R) |
TK |
Mobility Shift, IMAPTM |
08-155 |
FRK |
TK |
Mobility Shift, IMAPTM |
08-167 |
FYN |
TK |
Mobility Shift, IMAPTM |
08-068 |
GSK3α (GSK3A) |
STK |
Mobility Shift, IMAPTM |
04-140 |
GSK3β (GSK3B) |
STK |
Mobility Shift, IMAPTM |
04-141 |
Haspin (GSG2) |
STK |
Mobility Shift, IMAPTM |
05-111 |
HCK |
TK |
Mobility Shift, IMAPTM |
08-169 |
HER2 (ERBB2) |
TK |
Mobility Shift, IMAPTM |
08-016 |
HER4 (ERBB4) |
TK |
Mobility Shift, IMAPTM |
08-118 |
HGK (MAP4K4) |
STK |
Mobility Shift, IMAPTM |
07-137 |
HIPK1 |
STK |
Mobility Shift, IMAPTM |
04-135 |
HIPK2 |
STK |
Mobility Shift, IMAPTM |
04-136 |
HIPK3 |
STK |
Mobility Shift, IMAPTM |
04-137 |
HIPK4 |
STK |
Mobility Shift, IMAPTM |
04-138 |
IGF1R |
TK |
Mobility Shift, IMAPTM |
08-141 |
IKKα (CHUK) |
STK |
Mobility Shift, IMAPTM |
05-112 |
IKKβ (IKBKB) |
STK |
Mobility Shift, IMAPTM |
05-084 |
IKKε (IKBKE) |
STK |
Mobility Shift, IMAPTM |
05-114 |
INSR |
TK |
Mobility Shift, IMAPTM |
08-142 |
IRAK1 |
STK |
Mobility Shift, IMAPTM |
09-101 |
IRAK4 |
STK |
Mobility Shift, IMAPTM |
09-145 |
IRR (INSRR) |
TK |
Mobility Shift, IMAPTM |
08-143 |
ITK |
TK |
Mobility Shift, IMAPTM |
08-181 |
JAK1 |
TK |
Mobility Shift, IMAPTM |
08-144 |
JAK2 |
TK |
Mobility Shift, IMAPTM |
08-045 |
JAK3 |
TK |
Mobility Shift, IMAPTM |
08-046 |
JNK1 (MAPK8) |
STK |
Mobility Shift, IMAPTM |
04-163 |
JNK2 (MAPK9) |
STK |
Mobility Shift, IMAPTM |
04-164 |
JNK3 (MAPK10) |
STK |
Mobility Shift, IMAPTM |
04-150 |
KDR |
TK |
Mobility Shift, IMAPTM |
08-191 |
KIT |
TK |
Mobility Shift, IMAPTM |
08-156 |
KIT[D816V] |
TK |
Mobility Shift, IMAPTM |
08-505 |
KIT[T670I] |
TK |
Mobility Shift, IMAPTM |
08-195 |
KIT[V560G] |
TK |
Mobility Shift, IMAPTM |
08-504 |
KIT[V654A] |
TK |
Mobility Shift, IMAPTM |
08-511 |
LATS2 |
STK |
Mobility Shift, IMAPTM |
01-124 |
LCK |
TK |
Mobility Shift, IMAPTM |
08-170 |
LIMK1 |
STK |
ELISA |
09-105 |
LKB1(STK11)/MO25α/STRADα |
STK |
ELISA |
02-119 |
LOK (STK10) |
STK |
Mobility Shift, IMAPTM |
07-315 |
LTK |
TK |
Mobility Shift, IMAPTM |
08-106 |
LYNa |
TK |
Mobility Shift, IMAPTM |
08-171 |
LYNb |
TK |
Mobility Shift, IMAPTM |
08-172 |
MAP2K1 |
STK |
ELISA |
07-041 |
MAP2K1 |
STK |
Mobility Shift, IMAPTM |
07-141 |
MAP2K2 |
STK |
ELISA |
07-042 |
MAP2K2 |
STK |
Mobility Shift, IMAPTM |
07-142 |
MAP2K3 |
STK |
ELISA |
07-048 |
MAP2K3 |
STK |
Mobility Shift, IMAPTM |
07-143 |
MAP2K4 |
STK |
ELISA |
07-044 |
MAP2K4 |
STK |
Mobility Shift, IMAPTM |
07-144 |
MAP2K5 |
STK |
ELISA |
07-145 |
MAP2K5 |
STK |
Mobility Shift, IMAPTM |
07-145 |
MAP2K6 |
STK |
ELISA |
07-046 |
MAP2K6 |
STK |
Mobility Shift, IMAPTM |
07-146 |
MAP2K7 |
STK |
ELISA |
07-047 |
MAP2K7 |
STK |
Mobility Shift, IMAPTM |
07-148 |
MAP3K1 |
STK |
ELISA |
07-103 |
MAP3K1 |
STK |
Mobility Shift, IMAPTM |
07-103 |
MAP3K2 |
STK |
ELISA |
07-004 |
MAP3K2 |
STK |
Mobility Shift, IMAPTM |
07-104 |
MAP3K3 |
STK |
ELISA |
07-105 |
MAP3K3 |
STK |
Mobility Shift, IMAPTM |
07-105 |
MAP3K4 |
STK |
ELISA |
07-106 |
MAP3K4 |
STK |
Mobility Shift, IMAPTM |
07-106 |
MAP3K5 |
STK |
ELISA |
07-107 |
MAP3K5 |
STK |
Mobility Shift, IMAPTM |
07-107 |
MAP4K2 |
STK |
Mobility Shift, IMAPTM |
07-111 |
MAPKAPK2 |
STK |
Mobility Shift, IMAPTM |
02-142 |
MAPKAPK3 |
STK |
Mobility Shift, IMAPTM |
02-143 |
MAPKAPK5 |
STK |
Mobility Shift, IMAPTM |
02-144 |
MARK1 |
STK |
Mobility Shift, IMAPTM |
02-120 |
MARK2 |
STK |
Mobility Shift, IMAPTM |
02-121 |
MARK3 |
STK |
Mobility Shift, IMAPTM |
02-122 |
MARK4 |
STK |
Mobility Shift, IMAPTM |
02-123 |
MELK |
STK |
Mobility Shift, IMAPTM |
02-124 |
MER (MERTK) |
TK |
Mobility Shift, IMAPTM |
08-108 |
MET |
TK |
Mobility Shift, IMAPTM |
08-151 |
MET[Y1235D] |
TK |
Mobility Shift, IMAPTM |
08-198 |
MGC42105 |
STK |
Mobility Shift, IMAPTM |
02-125 |
MINK (MINK1) |
STK |
Mobility Shift, IMAPTM |
07-139 |
MLK1 (MAP3K9) |
STK |
Mobility Shift, IMAPTM |
09-115 |
MLK1(MAP3K9) |
STK |
ELISA |
09-015 |
MLK2 (MAP3K10) |
STK |
Mobility Shift, IMAPTM |
09-116 |
MLK2(MAP3K10) |
STK |
ELISA |
09-116 |
MLK3 (MAP3K11) |
STK |
Mobility Shift, IMAPTM |
09-017 |
MLK3(MAP3K11) |
STK |
ELISA |
09-017 |
MNK1 (MKNK1) |
STK |
Mobility Shift, IMAPTM |
02-145 |
MNK2 (MKNK2) |
STK |
Mobility Shift, IMAPTM |
02-146 |
MOS |
STK |
ELISA |
05-118 |
MOS |
STK |
Mobility Shift, IMAPTM |
05-118 |
MRCKα (CDC42BPA) |
STK |
Mobility Shift, IMAPTM |
01-107 |
MRCKβ (CDC42BPB) |
STK |
Mobility Shift, IMAPTM |
01-108 |
MSK1 (RPS6KA5) |
STK |
Mobility Shift, IMAPTM |
01-147 |
MSK2 (RPS6KA4) |
STK |
Mobility Shift, IMAPTM |
01-148 |
MSSK1 (STK23) |
STK |
Mobility Shift, IMAPTM |
04-159 |
MST1 (STK4) |
STK |
Mobility Shift, IMAPTM |
07-116 |
MST2 (STK3) |
STK |
Mobility Shift, IMAPTM |
07-117 |
MST3 (STK24) |
STK |
Mobility Shift, IMAPTM |
07-118 |
MST4 |
STK |
Mobility Shift, IMAPTM |
07-119 |
MUSK |
TK |
Mobility Shift, IMAPTM |
08-153 |
NDR1 (STK38) |
STK |
Mobility Shift, IMAPTM |
01-125 |
NDR2 (STK38L) |
STK |
Mobility Shift, IMAPTM |
01-126 |
NEK1 |
STK |
Mobility Shift, IMAPTM |
05-123 |
NEK2 |
STK |
Mobility Shift, IMAPTM |
05-226 |
NEK4 |
STK |
Mobility Shift, IMAPTM |
05-128 |
NEK6 |
STK |
Mobility Shift, IMAPTM |
05-130 |
NEK7 |
STK |
Mobility Shift, IMAPTM |
05-131 |
NEK9 |
STK |
Mobility Shift, IMAPTM |
05-133 |
NPM1-ALK |
TK |
Mobility Shift, IMAPTM |
08-517 |
NuaK1 |
STK |
Mobility Shift, IMAPTM |
02-126 |
NuaK2 |
STK |
Mobility Shift, IMAPTM |
02-127 |
p38α (MAPK14) |
STK |
Mobility Shift, IMAPTM |
04-152 |
p38β (MAPK11) |
STK |
Mobility Shift, IMAPTM |
04-153 |
p38γ (MAPK12) |
STK |
Mobility Shift, IMAPTM |
04-155 |
p38δ (MAPK13) |
STK |
Mobility Shift, IMAPTM |
04-154 |
p70S6K (RPS6KB1) |
STK |
Mobility Shift, IMAPTM |
01-154 |
p70S6Kβ (RPS6KB2) |
STK |
Mobility Shift, IMAPTM |
01-155 |
PAK1 |
STK |
Mobility Shift, IMAPTM |
07-123 |
PAK2 |
STK |
Mobility Shift, IMAPTM |
07-124 |
PAK3 |
STK |
Mobility Shift, IMAPTM |
07-125 |
PAK4 |
STK |
Mobility Shift, IMAPTM |
07-126 |
PAK5 (PAK7) |
STK |
Mobility Shift, IMAPTM |
07-127 |
PAK6 |
STK |
Mobility Shift, IMAPTM |
07-128 |
PASK |
STK |
Mobility Shift, IMAPTM |
02-128 |
PBK |
STK |
Mobility Shift, IMAPTM |
05-168 |
PDGFRα (PDGFRA) |
TK |
Mobility Shift, IMAPTM |
08-157 |
PDGFRα (PDGFRA) [T674I] |
TK |
Mobility Shift, IMAPTM |
08-503 |
PDGFRα (PDGFRA) [V561D] |
TK |
Mobility Shift, IMAPTM |
08-507 |
PDGFRβ (PDGFRB) |
TK |
Mobility Shift, IMAPTM |
08-158 |
PDHK2 (PDK2) |
STK |
Mobility Shift, IMAPTM |
10-140 |
PDHK4 (PDK4) |
STK |
Mobility Shift, IMAPTM |
10-125 |
PDK1 (PDPK1) |
STK |
Mobility Shift, IMAPTM |
01-132 |
PEK (EIF2AK3) |
STK |
Mobility Shift, IMAPTM |
05-155 |
PGK (PRKG1) |
STK |
Mobility Shift, IMAPTM |
01-142 |
PHKG1 |
STK |
Mobility Shift, IMAPTM |
02-152 |
PHKG2 |
STK |
Mobility Shift, IMAPTM |
02-153 |
PIK3CA/PIK3R1 |
Lipid |
Mobility Shift, IMAPTM |
11-101 |
PIM1 |
STK |
Mobility Shift, IMAPTM |
02-054 |
PIM2 |
STK |
Mobility Shift, IMAPTM |
02-155 |
PIM3 |
STK |
Mobility Shift, IMAPTM |
02-156 |
PKACα (PRKACA) |
STK |
Mobility Shift, IMAPTM |
01-127 |
PKACβ (PRKACB) |
STK |
Mobility Shift, IMAPTM |
01-128 |
PKACγ (PRKACG) |
STK |
Mobility Shift, IMAPTM |
01-129 |
PKCα (PRKCA) |
STK |
Mobility Shift, IMAPTM |
01-133 |
PKCβ1 (PRKCB1) |
STK |
Mobility Shift, IMAPTM |
01-134 |
PKCβ2 (PRKCB2) |
STK |
Mobility Shift, IMAPTM |
01-165 |
PKCγ (PRKCG) |
STK |
Mobility Shift, IMAPTM |
01-137 |
PKCδ (PRKCD) |
STK |
Mobility Shift, IMAPTM |
01-135 |
PKCε (PRKCE) |
STK |
Mobility Shift, IMAPTM |
01-136 |
PKCζ (PRKCZ) |
STK |
Mobility Shift, IMAPTM |
01-141 |
PKCη (PRKCH) |
STK |
Mobility Shift, IMAPTM |
01-138 |
PKCθ (PRKCQ) |
STK |
Mobility Shift, IMAPTM |
01-140 |
PKCι (PRKCI) |
STK |
Mobility Shift, IMAPTM |
01-139 |
PKD1 (PRKD1) |
STK |
Mobility Shift, IMAPTM |
02-157 |
PKD2 (PRKD2) |
STK |
Mobility Shift, IMAPTM |
02-158 |
PKD3 (PRKD3) |
STK |
Mobility Shift, IMAPTM |
02-159 |
PKN1 |
STK |
Mobility Shift, IMAPTM |
01-144 |
PKR (EIF2AK2) |
STK |
Mobility Shift, IMAPTM |
05-156 |
PLK1 |
STK |
Mobility Shift, IMAPTM |
05-157 |
PLK2 |
STK |
Mobility Shift, IMAPTM |
05-158 |
PLK3 |
STK |
Mobility Shift, IMAPTM |
05-159 |
PRKX |
STK |
Mobility Shift, IMAPTM |
01-130 |
PYK2 (PTK2B) |
TK |
Mobility Shift, IMAPTM |
08-138 |
QIK (SNF1LK2) |
STK |
Mobility Shift, IMAPTM |
02-129 |
RAF1 |
STK |
ELISA |
09-125 |
RAF1 |
STK |
Mobility Shift, IMAPTM |
09-125 |
RET |
TK |
Mobility Shift, IMAPTM |
08-159 |
RET[G691S] |
TK |
Mobility Shift, IMAPTM |
08-522 |
RET[M918T] |
TK |
Mobility Shift, IMAPTM |
08-508 |
RET[S891A] |
TK |
Mobility Shift, IMAPTM |
08-523 |
RET[Y791F] |
TK |
Mobility Shift, IMAPTM |
08-521 |
ROCK1 |
STK |
Mobility Shift, IMAPTM |
01-109 |
ROCK2 |
STK |
Mobility Shift, IMAPTM |
01-110 |
RON (MST1R) |
TK |
Mobility Shift, IMAPTM |
08-152 |
ROS (ROS1) |
TK |
Mobility Shift, IMAPTM |
08-163 |
RSK1 (RPS6KA1) |
STK |
Mobility Shift, IMAPTM |
01-149 |
RSK2 (RPS6KA3) |
STK |
Mobility Shift, IMAPTM |
01-150 |
RSK3 (RPS6KA2) |
STK |
Mobility Shift, IMAPTM |
01-151 |
RSK4 (RPS6KA6) |
STK |
Mobility Shift, IMAPTM |
01-152 |
SGK |
STK |
Mobility Shift, IMAPTM |
01-158 |
SGK2 |
STK |
Mobility Shift, IMAPTM |
01-159 |
SGK3 (SGKL) |
STK |
Mobility Shift, IMAPTM |
01-160 |
SIK (SNF1LK) |
STK |
Mobility Shift, IMAPTM |
02-131 |
skMLCK (MYLK2) |
STK |
Mobility Shift, IMAPTM |
02-150 |
SLK |
STK |
Mobility Shift, IMAPTM |
07-129 |
SPHK1 |
Lipid |
Mobility Shift, IMAPTM |
11-105 |
SPHK2 |
Lipid |
Mobility Shift, IMAPTM |
11-106 |
SRC |
TK |
Mobility Shift, IMAPTM |
08-173 |
SRM (SRMS) |
TK |
Mobility Shift, IMAPTM |
08-174 |
SRPK1 |
STK |
Mobility Shift, IMAPTM |
04-160 |
SRPK2 |
STK |
Mobility Shift, IMAPTM |
04-161 |
SYK |
TK |
Mobility Shift, IMAPTM |
08-176 |
TAK1-TAB1 (MAP3K7) |
STK |
Mobility Shift, IMAPTM |
09-019 |
TAK1-TAB1(MAP3K7) |
STK |
ELISA |
09-019 |
TAOK2 |
STK |
Mobility Shift, IMAPTM |
07-133 |
TBK1 |
STK |
Mobility Shift, IMAPTM |
05-115 |
TEC |
TK |
Mobility Shift, IMAPTM |
08-182 |
TIE2 (TEK) |
TK |
Mobility Shift, IMAPTM |
08-185 |
TNIK |
STK |
Mobility Shift, IMAPTM |
07-138 |
TNK1 |
TK |
Mobility Shift, IMAPTM |
08-104 |
TRKA (NTRK1) |
TK |
Mobility Shift, IMAPTM |
08-186 |
TRKB (NTRK2) |
TK |
Mobility Shift, IMAPTM |
08-187 |
TRKC (NTRK3) |
TK |
Mobility Shift, IMAPTM |
08-197 |
TSSK1 |
STK |
Mobility Shift, IMAPTM |
02-364 |
TSSK2 |
STK |
Mobility Shift, IMAPTM |
02-165 |
TSSK3 |
STK |
Mobility Shift, IMAPTM |
02-166 |
TTK |
STK |
ELISA |
05-169 |
TXK |
TK |
Mobility Shift, IMAPTM |
08-183 |
TYK2 |
TK |
Mobility Shift, IMAPTM |
08-147 |
TYRO3 |
TK |
Mobility Shift, IMAPTM |
08-109 |
WEE1 |
STK |
ELISA |
05-177 |
WNK1 |
STK |
Mobility Shift, IMAPTM |
05-179 |
WNK2 |
STK |
Mobility Shift, IMAPTM |
05-180 |
WNK3 |
STK |
Mobility Shift, IMAPTM |
05-181 |
YES (YES1) |
TK |
Mobility Shift, IMAPTM |
08-175 |
YES (YES1) [T348I] |
TK |
Mobility Shift, IMAPTM |
08-533 |
High [ATP] Kinase Panel
Through our partner Carna Biosciences we are offering the high [ATP] kinase panel. This panel facilitates inhibitor-type determinations (type I, II or III) by adding optional profiling at 1 mM ATP and kinase selectivity at physiological ATP levels.
Kinases Available in the high [ATP] kinase panel
The high ATP kinase panel comprises 166 human kinases (107 TKs including mutants, 59 STKs) and allows the impact of ATP concentration on kinase-inhibitory activity to be rapidly visualized and assessed. Despite the sensitivity offered by performing in vitro assays at ATP concentrations approximating Km, physiological conditions are seldom the same. Inhibitory potency and selectivity may vary with the concentration of ATP available.
Target Name | Group |
Source (Carna Cat No.) |
ABL (ABL1) | TK | 08-001 |
ABL (ABL1) [T315I] | TK | 08-093 |
ABL (ABL1) [E255K] | TK | 08-094 |
ACK (TNK2) | TK | 08-196 |
AKT1 | STK | 01-101 |
ALK | TK | 08-518 |
ALK[F1174L] | TK | 08-519 |
ALK[L1196M] | TK | 08-529 |
ALK[R1275Q] | TK | 08-520 |
AMPK α1/β1/γ1 (PRKAA1/B1/G1) | STK | 02-113 |
ARG (ABL2) | TK | 08-102 |
AurA (AURKA) | STK | 05-101 |
AurB (AURKB)/INCENP | STK | 05-102 |
AurC (AURKC) | STK | 05-103 |
AXL | TK | 08-107 |
BLK | TK | 08-164 |
BMX | TK | 08-179 |
BRK (PTK6) | TK | 08-165 |
BRSK1 | STK | 02-115 |
BTK | TK | 08-080 |
CaMK4 | STK | 02-108 |
CDC2 /CycB1 | STK | 04-102 |
CDC7/ASK | STK | 05-109 |
CDK2 /CycE1 | STK | 04-165 |
CDK2 /CycA2 | STK | 04-103 |
CDK4 /CycD3 | STK | 04-105 |
CDK5 /p25 | STK | 04-106 |
CDK6 /CycD3 | STK | 04-107 |
CDK7 /CycH/MAT1 | STK | 04-108 |
CDK9 /CycT1 | STK | 04-110 |
CHK1 (CHEK1) | STK | 02-117 |
CHK2 (CHEK2) | STK | 02-162 |
CK1α (CSNK1A1) | STK | 03-101 |
CK1ε (CSNK1E) | STK | 03-104 |
CK2α1/β (CSNK2A1/B) | STK | 05-184 |
CSK | TK | 08-111 |
DAPK1 | STK | 02-134 |
DDR1 | TK | 08-113 |
DDR2 | TK | 08-114 |
DYRK1B | STK | 04-131 |
EGFR | TK | 08-115 |
EGFR[d746-750/T790M] | TK | 08-528 |
EGFR[d746-750] | TK | 08-527 |
EGFR[L858R] | TK | 08-502 |
EGFR[L861Q] | TK | 08-513 |
EGFR[T790M/L858R] | TK | 08-510 |
EGFR[T790M] | TK | 08-194 |
EML4-ALK | TK | 08-516 |
EPHA1 | TK | 08-119 |
EPHA2 | TK | 08-121 |
EPHA3 | TK | 08-122 |
EPHA4 | TK | 08-123 |
EPHA5 | TK | 08-124 |
EPHA6 | TK | 08-125 |
EPHA7 | TK | 08-126 |
EPHA8 | TK | 08-127 |
EPHB1 | TK | 08-128 |
EPHB2 | TK | 08-129 |
EPHB3 | TK | 08-130 |
EPHB4 | TK | 08-131 |
Erk1 (MAPK3) | STK | 04-142 |
Erk2 (MAPK1) | STK | 04-143 |
FAK (PTK2) | TK | 08-137 |
FER | TK | 08-139 |
FES | TK | 08-140 |
FGFR1 | TK | 08-133 |
FGFR2 | TK | 08-134 |
FGFR3 | TK | 08-135 |
FGFR3[K650E] | TK | 08-501 |
FGFR3[K650M] | TK | 08-199 |
FGFR4 | TK | 08-136 |
FGFR4[N535K] | TK | 08-524 |
FGFR4[V550E] | TK | 08-525 |
FGFR4[V550L] | TK | 08-526 |
FGR | TK | 08-166 |
FLT1 | TK | 08-189 |
FLT3 | TK | 08-154 |
FLT4 | TK | 08-190 |
FMS (CSF1R) | TK | 08-155 |
FRK | TK | 08-167 |
FYN | TK | 08-068 |
GSK3α (GSK3A) | STK | 04-140 |
GSK3β (GSK3B) | STK | 04-141 |
HCK | TK | 08-169 |
HER2 (ERBB2) | TK | 08-016 |
HER4 (ERBB4) | TK | 08-118 |
HGK (MAP4K4) | STK | 07-137 |
IGF1R | TK | 08-141 |
IKKβ (IKBKB) | STK | 05-084 |
INSR | TK | 08-142 |
IRR (INSRR) | TK | 08-143 |
ITK | TK | 08-181 |
JAK1 | TK | 08-144 |
JAK2 | TK | 08-045 |
JAK3 | TK | 08-046 |
JNK1 (MAPK8) | STK | 04-163 |
JNK2 (MAPK9) | STK | 04-164 |
JNK3 (MAPK10) | STK | 04-150 |
KDR | TK | 08-191 |
KIT | TK | 08-156 |
KIT[D816V] | TK | 08-505 |
KIT[T670I] | TK | 08-195 |
KIT[V560G] | TK | 08-504 |
KIT[V654A] | TK | 08-511 |
LCK | TK | 08-170 |
LTK | TK | 08-106 |
LYNa | TK | 08-171 |
LYNb | TK | 08-172 |
MAPKAPK2 | STK | 02-142 |
MER (MERTK) | TK | 08-108 |
MET | TK | 08-151 |
MET[Y1235D] | TK | 08-198 |
MST1 (STK4) | STK | 07-116 |
MUSK | TK | 08-153 |
NEK1 | STK | 05-123 |
NEK2 | STK | 05-226 |
NEK6 | STK | 05-130 |
NEK7 | STK | 05-131 |
NEK9 | STK | 05-133 |
NPM1-ALK | TK | 08-517 |
p38α (MAPK14) | STK | 04-152 |
p38β (MAPK11) | STK | 04-153 |
p38γ (MAPK12) | STK | 04-155 |
p38δ (MAPK13) | STK | 04-154 |
p70S6K (RPS6KB1) | STK | 01-154 |
PAK2 | STK | 07-124 |
PBK | STK | 05-168 |
PDGFRα (PDGFRA) | TK | 08-157 |
PDGFRα (PDGFRA) [T674I] | TK | 08-503 |
PDGFRα (PDGFRA) [V561D] | TK | 08-507 |
PDGFRβ (PDGFRB) | TK | 08-158 |
PDK1 (PDPK1) | STK | 01-132 |
PIM1 | STK | 02-054 |
PIM2 | STK | 02-155 |
PKACα (PRKACA) | STK | 01-127 |
PKCα (PRKCA) | STK | 01-133 |
PKCε (PRKCE) | STK | 01-136 |
PKD2 (PRKD2) | STK | 02-158 |
PLK1 | STK | 05-157 |
PLK3 | STK | 05-159 |
PYK2 (PTK2B) | TK | 08-138 |
RET | TK | 08-159 |
RET[G691S] | TK | 08-522 |
RET[M918T] | TK | 08-508 |
RET[S891A] | TK | 08-523 |
RET[Y791F] | TK | 08-521 |
ROCK1 | STK | 01-109 |
RON (MST1R) | TK | 08-152 |
ROS (ROS1) | TK | 08-163 |
RSK1 (RPS6KA1) | STK | 01-149 |
SGK | STK | 01-158 |
SRC | TK | 08-173 |
SRM (SRMS) | TK | 08-174 |
SYK | TK | 08-176 |
TEC | TK | 08-182 |
TIE2 (TEK) | TK | 08-185 |
TNK1 | TK | 08-104 |
TRKA (NTRK1) | TK | 08-186 |
TRKB (NTRK2) | TK | 08-187 |
TRKC (NTRK3) | TK | 08-197 |
TSSK1 | STK | 02-364 |
TXK | TK | 08-183 |
TYK2 | TK | 08-147 |
TYRO3 | TK | 08-109 |
YES (YES1) | TK | 08-175 |
QuickScout™ Cell Cycle Panel
Through our partner Carna Biosciences we are offering QuickScout™ Cell Cycle Panel v2.0. This panel is comprised of relevant kinases for cell-cycle regulation and best for determining whether your compound acts on cell multiplication.
Kinases Available in QuickScout™ Cell Cycle panel
The QuickScout™ Cell Cycle Panel mainly includes kinases which are directly involved in the cell-cycle, and their inhibition may interfere with cell proliferation. Contact us to learn more about this panel and how we can help you identify the clinical potential of your compounds.
Target Name | Group |
Source (Carna Cat No.) |
AurA (AURKA) | STK | 05-101 |
AurB (AURKB)/INCENP | STK | 05-102 |
AurC (AURKC) | STK | 05-103 |
BRSK2 | STK | 02-116 |
CDC2 /CycB1 | STK | 04-102 |
CDC7/ASK | STK | 05-109 |
CDK2 /CycE1 | STK | 04-165 |
CDK2 /CycA2 | STK | 04-103 |
CDK3 /CycE1 | STK | 04-104 |
CDK4 /CycD3 | STK | 04-105 |
CDK6 /CycD3 | STK | 04-107 |
CDK7 /CycH/MAT1 | STK | 04-108 |
CDK9 /CycT1 | STK | 04-110 |
CHK1 (CHEK1) | STK | 02-117 |
CHK2 (CHEK2) | STK | 02-162 |
CK2 α1/β (CSNK2A1/B) | STK | 05-184 |
CK2 α2/β (CSNK2A2/B) | STK | 05-185 |
GSK3 β (GSK3B) | STK | 04-141 |
NEK1 | STK | 05-123 |
NEK2 | STK | 05-226 |
NEK6 | STK | 05-130 |
NEK7 | STK | 05-131 |
NEK9 | STK | 05-133 |
p38 α (MAPK14) | STK | 04-152 |
p70S6K (RPS6KB1) | STK | 01-154 |
PIM1 | STK | 02-054 |
PIM2 | STK | 02-155 |
PLK1 | STK | 05-157 |
PLK2 | STK | 05-158 |
RSK1 (RPS6KA1) | STK | 01-149 |
QuickScout™ STK Panel
Through our partner Carna Biosciences we are offering the QuickScout™ STK Panel v2.0. This panel of 30 pre-selected Serine/Threonine kinases is comprised of key members from the AGC, CAMK, CMGC, STE, TKL, and Other Group of STK kinases.
Kinases Available in QuickScout™ STK panel
This panel allows you to screen your lead compounds using the industry’s most diverse Kinome Sampler and helps you discover and characterize the selectivity of your compounds as potential treatments for cancer, inflammatory, metabolic and/or neurological diseases. Contact us to learn more about this panel and how we can help you identify the clinical potential of your compounds.
Target Name | Group |
Source (Carna Cat No.) |
AKT1 | STK | 01-101 |
AMPKα1/β1/γ1 (PRKAA1/B1/G1) | STK | 02-113 |
AurA (AURKA) | STK | 05-101 |
CaMK4 | STK | 02-108 |
CDK2 /CycA2 | STK | 04-103 |
CHK1 (CHEK1) | STK | 02-117 |
CK1ε (CSNK1E) | STK | 03-104 |
DAPK1 | STK | 02-134 |
DYRK1B | STK | 04-131 |
Erk2 (MAPK1) | STK | 04-143 |
GSK3β (GSK3B) | STK | 04-141 |
HGK (MAP4K4) | STK | 07-137 |
IKKβ (IKBKB) | STK | 05-084 |
IRAK4 | STK | 09-145 |
JNK2 (MAPK9) | STK | 04-164 |
MAPKAPK2 | STK | 02-142 |
MST1 (STK4) | STK | 07-116 |
NEK2 | STK | 05-226 |
p38α (MAPK14) | STK | 04-152 |
p70S6K (RPS6KB1) | STK | 01-154 |
PAK2 | STK | 07-124 |
PBK | STK | 05-168 |
PDK1 (PDPK1) | STK | 01-132 |
PIM1 | STK | 02-054 |
PKACα (PRKACA) | STK | 01-127 |
PKCα (PRKCA) | STK | 01-133 |
PKD2 (PRKD2) | STK | 02-158 |
ROCK1 | STK | 01-109 |
SGK | STK | 01-158 |
TSSK1 | STK | 02-364 |
QuickScout™ TK Panel
Through our partner Carna Biosciences we are offering the QuickScout™ TK Panel v2.0. This panel of 20 pre-selected Tyrosine Kinases (TKs) is comprised of both receptor and non-receptor TKs and is offered to help you to rapidly screen your compounds against druggable and clinically relevant kinases.
Kinases Available in QuickScout™ TK panel
Identification and optimization of small molecular inhibitors against many of the targets in our 20 TK panel has led to the development of first and second generation therapeutics for the treatment of diseases such as leukemia and cancers of the lung, breast, and kidney. Contact us to learn more about this Panel and how we can help you identify the clinical potential of your compounds.
Target Name | Group |
Source (Carna Cat No.) |
ABL (ABL1) | TK | 08-001 |
CSK | TK | 08-111 |
EGFR | TK | 08-115 |
EPHA2 | TK | 08-121 |
EPHB4 | TK | 08-131 |
FGFR1 | TK | 08-133 |
FLT3 | TK | 08-154 |
IGF1R | TK | 08-141 |
ITK | TK | 08-181 |
JAK3 | TK | 08-046 |
KDR | TK | 08-191 |
LCK | TK | 08-170 |
MET | TK | 08-151 |
PDGFR α (PDGFRA) | TK | 08-157 |
PYK2 (PTK2B) | TK | 08-138 |
SRC | TK | 08-173 |
SYK | TK | 08-176 |
TIE2 (TEK) | TK | 08-185 |
TRKA (NTRK1) | TK | 08-186 |
TYRO3 | TK | 08-109 |